Oxybutynin chloride
Modify Date: 2024-01-09 13:25:50
Oxybutynin chloride structure
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Common Name | Oxybutynin chloride | ||
|---|---|---|---|---|
| CAS Number | 1508-65-2 | Molecular Weight | 393.947 | |
| Density | N/A | Boiling Point | 494.4ºC at 760 mmHg | |
| Molecular Formula | C22H32ClNO3 | Melting Point | 126-128ºC | |
| MSDS | Chinese USA | Flash Point | N/A | |
| Symbol |
GHS07 |
Signal Word | Warning | |
Use of Oxybutynin chlorideOxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties.Target: mAChROxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties, including frequent urination and inability to control urination (urge incontinence), by decreasing muscle spasms of the bladder. Oxybutynin competitively antagonizes the M1, M2, and M3 subtypes of the muscarinic acetylcholine receptor. It also has direct spasmolytic effects on bladder smooth muscle as a calcium antagonist and local anesthetic, but at concentrations far above those used clinically. Oxybutynin is available orally in generic formulation or as the brand-names Ditropan, Lyrinel XL, or Ditrospam, as a transdermal patch under the brand name Oxytrol, and as a topical gel under the brand name Gelnique. Oxybutynin is also a possible treatment of hyperhidrosis (hyper-active sweating) [1-3]. |
| Name | oxybutynin chloride |
|---|---|
| Synonym | More Synonyms |
| Description | Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties.Target: mAChROxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties, including frequent urination and inability to control urination (urge incontinence), by decreasing muscle spasms of the bladder. Oxybutynin competitively antagonizes the M1, M2, and M3 subtypes of the muscarinic acetylcholine receptor. It also has direct spasmolytic effects on bladder smooth muscle as a calcium antagonist and local anesthetic, but at concentrations far above those used clinically. Oxybutynin is available orally in generic formulation or as the brand-names Ditropan, Lyrinel XL, or Ditrospam, as a transdermal patch under the brand name Oxytrol, and as a topical gel under the brand name Gelnique. Oxybutynin is also a possible treatment of hyperhidrosis (hyper-active sweating) [1-3]. |
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| Related Catalog | |
| References |
| Boiling Point | 494.4ºC at 760 mmHg |
|---|---|
| Melting Point | 126-128ºC |
| Molecular Formula | C22H32ClNO3 |
| Molecular Weight | 393.947 |
| Exact Mass | 393.207062 |
| PSA | 49.77000 |
| LogP | 4.14490 |
| Vapour Pressure | 1.37E-10mmHg at 25°C |
| Storage condition | Room temp |
CHEMICAL IDENTIFICATION
HEALTH HAZARD DATAACUTE TOXICITY DATA
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| Symbol |
GHS07 |
|---|---|
| Signal Word | Warning |
| Hazard Statements | H302 |
| Precautionary Statements | P301 + P312 + P330 |
| Personal Protective Equipment | dust mask type N95 (US);Eyeshields;Faceshields;Gloves |
| Hazard Codes | Xn |
| Risk Phrases | R22 |
| Safety Phrases | 36 |
| RIDADR | NONH for all modes of transport |
| RTECS | GV2800000 |
| HS Code | 2921590090 |
| Precursor 0 | |
|---|---|
| DownStream 3 | |
CAS#:5633-20-5
CAS#:10575-25-4
CAS#:4335-77-7| HS Code | 2922509090 |
|---|---|
| Summary | 2922509090. other amino-alcohol-phenols, amino-acid-phenols and other amino-compounds with oxygen function. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:30.0% |
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| EINECS 216-139-7 |
| a-Cyclohexyl-a-hydroxybenzeneacetic Acid 4-(Diethylamino)-2-butynyl Ester Hydrochloride |
| a-Phenylcyclohexaneglycolic Acid 4-(Diethylamino)-2-butynyl Ester Hydrochloride |
| Oxybutynin hydrochloride |
| Oxybutynin Chloride |
| benzeneacetic acid, a-cyclohexyl-a-hydroxy-, 4-(diethylamino)-2-butyn-1-yl ester, hydrochloride (1:1) |
| 4-(Diethylamino)but-2-in-1-ylcyclohexyl(hydroxy)phenylacetathydrochlorid |
| MFCD00072150 |
| 4-(Diethylamino)but-2-yn-1-yl cyclohexyl(hydroxy)phenylacetate hydrochloride (1:1) |
| cyclohexyl(hydroxy)phénylacétate de 4-(diéthylamino)but-2-yn-1-yle chlorhydrate |
| Benzeneacetic acid, α-cyclohexyl-α-hydroxy-, 4-(diethylamino)-2-butyn-1-yl ester, hydrochloride (1:1) |
| 4-Diethylamino-2-butynyl Phenylcyclohexylglycolate Hydrochloride |
| benzeneacetic acid, α-cyclohexyl-α-hydroxy-, 4-(diethylamino)-2-butynyl ester, hydrochloride |
| 4-(Diethylamino)-2-butyn-1-yl cyclohexyl(hydroxy)phenylacetate hydrochloride (1:1) |
| 4-{[cyclohexyl(hydroxy)phenylacetyl]oxy}-N,N-diethylbut-2-yn-1-aminium chloride |
| Oxybutynin HCl |