DC-TEADin1072

Modify Date: 2024-04-05 19:01:28

DC-TEADin1072 Structure
DC-TEADin1072 structure
 Common Name DC-TEADin1072
CAS Number 1574602-93-9 Molecular Weight 259.349
Density N/A Boiling Point N/A
Molecular Formula C16H21NO2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of DC-TEADin1072


DC-TEADin1072 is a novel TEAD1/3 covalent inhibitor with biochemical IC50 values of 0.61 and 0.58 uM against TEAD1 and TEAD3, respectively.TEADin1072 selectively inhibited TEAD1 and TEAD3 palmitoylation while sparing TEAD2 and TEAD4.TEADin1072 demonstrated selective engagement with Cys371 of TEAD3 and Cys359 of TEAD1.

 Names

Name DC-TEADin1072

 DC-TEADin1072 Biological Activity

Description DC-TEADin1072 is a novel TEAD1/3 covalent inhibitor with biochemical IC50 values of 0.61 and 0.58 uM against TEAD1 and TEAD3, respectively.TEADin1072 selectively inhibited TEAD1 and TEAD3 palmitoylation while sparing TEAD2 and TEAD4.TEADin1072 demonstrated selective engagement with Cys371 of TEAD3 and Cys359 of TEAD1.
References 1. Tian Lu, et al. Acta Pharm Sin B. 2021 Oct;11(10):3206-3219.

 Chemical & Physical Properties

Molecular Formula C16H21NO2
Molecular Weight 259.349
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Chemsrc provides DC-TEADin1072(CAS#:1574602-93-9) MSDS, density, melting point, boiling point, structure, formula, molecular weight etc. Articles of DC-TEADin1072 are included as well.>> amp version: DC-TEADin1072

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