Mambalgin 1
Modify Date: 2024-01-12 22:42:42
Mambalgin 1 structure
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Common Name | Mambalgin 1 | ||
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| CAS Number | 1609937-15-6 | Molecular Weight | 7283.22 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C310H481N87O100S8 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Mambalgin 1Mambalgin 1 is a selective ASIC1a inhibitor (IC50 values are 192 and 72 nM for human ASIC1a and ASIC1a/1b dimer, respectively). Mambalgin 1 binds to closed/inactive channel. Mambalgin 1 is selective for ASIC1a over ASIC2a, ASIC3, TRPV1, P2X2, 5-HT3, Nav1.8, Cav3.2 and Kv1.2 channels. Mambalgin 1 increases latency of withdrawal response in mouse tail-flick and paw-flick tests. |
| Name | Mambalgin 1 |
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| Description | Mambalgin 1 is a selective ASIC1a inhibitor (IC50 values are 192 and 72 nM for human ASIC1a and ASIC1a/1b dimer, respectively). Mambalgin 1 binds to closed/inactive channel. Mambalgin 1 is selective for ASIC1a over ASIC2a, ASIC3, TRPV1, P2X2, 5-HT3, Nav1.8, Cav3.2 and Kv1.2 channels. Mambalgin 1 increases latency of withdrawal response in mouse tail-flick and paw-flick tests. |
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| Related Catalog |
| Molecular Formula | C310H481N87O100S8 |
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| Molecular Weight | 7283.22 |