ZEN-3694

Modify Date: 2024-09-22 17:36:29

ZEN-3694 Structure
ZEN-3694 structure
Common Name ZEN-3694
CAS Number 1643947-30-1 Molecular Weight 333.39
Density N/A Boiling Point N/A
Molecular Formula C19H19N5O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of ZEN-3694


ZEN-3694 is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and can be used in combination with enzalutamide to study metastatic desmoplasia-resistant prostate cancer.

 Names

Name ZEN-3694

 ZEN-3694 Biological Activity

Description ZEN-3694 is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and can be used in combination with enzalutamide to study metastatic desmoplasia-resistant prostate cancer.
References 1. Aggarwal RR, et al. A Phase Ib/IIa Study of the Pan-BET Inhibitor ZEN-3694 in Combination with Enzalutamide in Patients with Metastatic Castration-resistant Prostate Cancer. Clin Cancer Res. 2020 Oct 15;26(20):5338-5347.

 Chemical & Physical Properties

Molecular Formula C19H19N5O
Molecular Weight 333.39
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.