1643947-30-1
1643947-30-1 structure
- Name: ZEN-3694
- Chemical Name: ZEN-3694
- CAS Number: 1643947-30-1
- Molecular Formula: C19H19N5O
- Molecular Weight: 333.39
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2024-09-22 17:36:29
- Modify Date: 2025-08-25 16:59:19
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ZEN-3694 is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and can be used in combination with enzalutamide to study metastatic desmoplasia-resistant prostate cancer.
| Name | ZEN-3694 |
|---|
| Description | ZEN-3694 is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and can be used in combination with enzalutamide to study metastatic desmoplasia-resistant prostate cancer. |
|---|---|
| References | 1. Aggarwal RR, et al. A Phase Ib/IIa Study of the Pan-BET Inhibitor ZEN-3694 in Combination with Enzalutamide in Patients with Metastatic Castration-resistant Prostate Cancer. Clin Cancer Res. 2020 Oct 15;26(20):5338-5347. |
| Molecular Formula | C19H19N5O |
|---|---|
| Molecular Weight | 333.39 |