PD 168568 dihydrochloride
Modify Date: 2024-01-17 20:31:25
PD 168568 dihydrochloride structure
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Common Name | PD 168568 dihydrochloride | ||
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| CAS Number | 1782532-06-2 | Molecular Weight | 422.39 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C22H29Cl2N3O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PD 168568 dihydrochloridePD 168568 dihydrochloride is an orally active and selective D4 dopamine receptor antagonist, with a Ki of 8.8 nM[1]. |
| Name | PD 168568 dihydrochloride |
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| Description | PD 168568 dihydrochloride is an orally active and selective D4 dopamine receptor antagonist, with a Ki of 8.8 nM[1]. |
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| Related Catalog | |
| Target |
D4 Receptor:8.8 nM (Ki) |
| In Vitro | PD 168568 dihydrochloride has good selective for D4 receptor, with a Ki of 1842 nM for D2 receptor[1]. |
| In Vivo | PD 168568 dihydrochloride has ability to inhibit amphetamine stimulated locomotor activity in the rat[1]. Animal Model: Rat[1] Dosage: 3 mg/kg Administration: Oral administration Result: Inhibit amphetamine (0.5 mg/kg, i.p.) stimulated locomotor activity. |
| References |
| Molecular Formula | C22H29Cl2N3O |
|---|---|
| Molecular Weight | 422.39 |
| Storage condition | 2-8°C |