MRS1177

Modify Date: 2024-01-14 00:28:30

MRS1177 structure	Common Name	MRS1177
	CAS Number	183721-13-3	Molecular Weight	389.79
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₀H₁₂ClN₅O₂	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of MRS1177

MRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM.

Name	MRS1177

Description	MRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Adenosine Receptor Research Areas >> Others
Target	Ki: 0.3 nM (hA3AR)[1][2].
In Vitro	MRS1177 (compound 2b) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist[1]. The Ki value of MRS1177 (compound 55) with hA3AR is 0.3 nM[2].
References	[1]. Tafi A, et al. Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models. J Med Chem. 2006 Jul 13;49(14):4085-97. [2]. Cheong SL, et al. Pharmacophore elucidation for a new series of 2-aryl-pyrazolo-triazolo-pyrimidines as potent human A3 adenosine receptor antagonists. Bioorg Med Chem Lett. 2011 May 15;21(10):2898-905.

Molecular Formula	C₂₀H₁₂ClN₅O₂
Molecular Weight	389.79

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China
Product Name: MRS1177
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DC Chemicals Limited
China
Product Name: MRS1177
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ShangHai DC Chemicals Co.,Ltd
China
Product Name: MRS1177
Price: ￥Inquiry/1g
Purity: 98.9%
Delivery: 1 Day
Contact: Tony Lai
Email: order@dcchemicals.com

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