ML233
Modify Date: 2024-01-08 09:51:45
ML233 structure
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Common Name | ML233 | ||
|---|---|---|---|---|
| CAS Number | 2080311-92-6 | Molecular Weight | 359.44 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C19H21NO4S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of ML233ML233 is a non-peptide based potent apelin receptor (APJ) agonist (EC50=3.7 μM). ML233 displays >21-fold selective over the closely related angiotensin 1 (AT1) receptor (>79 μM)[1]. |
| Name | ML233 |
|---|
| Description | ML233 is a non-peptide based potent apelin receptor (APJ) agonist (EC50=3.7 μM). ML233 displays >21-fold selective over the closely related angiotensin 1 (AT1) receptor (>79 μM)[1]. |
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| Related Catalog | |
| Target |
EC50: 3.7 μM (Apelin receptor)[1] |
| In Vitro | ML233 shows potentially significant binding against several other receptors, including the 5-HT1A, α2C adrenergic, and benzylpiperazine receptors and norepinephrine transporter. ML233 shows some toxicity (LC50=25.8 μM) toward human hepatocyctes[1]. |
| References |
| Molecular Formula | C19H21NO4S |
|---|---|
| Molecular Weight | 359.44 |