VCP-Eribulin

Modify Date: 2024-01-09 19:08:14

VCP-Eribulin Structure
VCP-Eribulin structure
Common Name VCP-Eribulin
CAS Number 2130869-17-7 Molecular Weight 1135.34
Density N/A Boiling Point N/A
Molecular Formula C59H86N6O16 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of VCP-Eribulin


VCP-Eribulin consists the ADCs linker (VCP) and Eribulin[1]. Eribulin is a mechanistically unique microtubule inhibitor for cancer[2]. VCP-Eribulin is an Eribulin-based drug for antibody conjugates[1].

 Names

Name VCP-Eribulin

 VCP-Eribulin Biological Activity

Description VCP-Eribulin consists the ADCs linker (VCP) and Eribulin[1]. Eribulin is a mechanistically unique microtubule inhibitor for cancer[2]. VCP-Eribulin is an Eribulin-based drug for antibody conjugates[1].
Related Catalog
References

[1]. Earl F Albone, et al. Eribulin-based antibody-drug conjugates and methods of use. US20170252458A1.

[2]. Towle MJ, et al. Eribulin induces irreversible mitotic blockade: implications of cell-based pharmacodynamics for in vivo efficacy under intermittent dosing conditions. Cancer Res. 2011 Jan 15;71(2):496-505.

 Chemical & Physical Properties

Molecular Formula C59H86N6O16
Molecular Weight 1135.34
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