RJR 2403 oxalate

Modify Date: 2024-01-02 18:44:37

RJR 2403 oxalate structure	Common Name	RJR 2403 oxalate
	CAS Number	220662-95-3	Molecular Weight	252.26600
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₁₂H₁₆N₂O₄	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of RJR 2403 oxalate

Rivanicline oxalate (RJR-2403 oxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 36000 nM).

Name	(E)-N-methyl-4-pyridin-3-ylbut-3-en-1-amine,oxalic acid
Synonym	More Synonyms

Description	Rivanicline oxalate (RJR-2403 oxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 36000 nM).
Related Catalog	Signaling Pathways >> Membrane Transporter/Ion Channel >> nAChR Signaling Pathways >> Neuronal Signaling >> nAChR Research Areas >> Neurological Disease
References	[1]. Bencherif M, et al. RJR-2403: a nicotinic agonist with CNS selectivity I. In vitro characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1413-21. [2]. Lippiello PM, et al. RJR-2403: a nicotinic agonist with CNS selectivity II. In vivo characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1422-9. [3]. Damaj MI, et al. Antinociceptive and pharmacological effects of metanicotine, a selective nicotinic agonist. J Pharmacol Exp Ther. 1999 Oct;291(1):390-8.

Description

Rivanicline oxalate (RJR-2403 oxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 36000 nM).

Related Catalog

Signaling Pathways >> Membrane Transporter/Ion Channel >> nAChR

Signaling Pathways >> Neuronal Signaling >> nAChR

Research Areas >> Neurological Disease

References

[1]. Bencherif M, et al. RJR-2403: a nicotinic agonist with CNS selectivity I. In vitro characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1413-21.

[2]. Lippiello PM, et al. RJR-2403: a nicotinic agonist with CNS selectivity II. In vivo characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1422-9.

[3]. Damaj MI, et al. Antinociceptive and pharmacological effects of metanicotine, a selective nicotinic agonist. J Pharmacol Exp Ther. 1999 Oct;291(1):390-8.

Molecular Formula	C₁₂H₁₆N₂O₄
Molecular Weight	252.26600
Exact Mass	252.11100
PSA	99.52000
LogP	1.25080
Storage condition	2-8℃

Rivanicline oxalate

CS-0531

RJR-2403 oxalate

RJR-2403 oxalate||Rivanicline oxalate|RJR 2403 oxalate

RJR-2403 (oxalate)

DC Chemicals Limited
China
Product Name: RJR-2403 oxalate
Price: $Inquiry/10mg $Inquiry/25mg $Inquiry/50mg
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

Dayang Chem (Hangzhou) Co., Ltd.
China
Product Name: RJR-2403 (oxalate)
Price: $Inquiry/100g $Inquiry/1kg $Inquiry/100kg $Inquiry/1000kg
Purity: 98.0%
Stocking Period: Inquiry
Contact: Ms Wang

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Price: $132/10mg

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RJR 2403 oxalate

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