(Rac)-CP-601927 hydrochloride

Modify Date: 2024-01-03 11:31:17

(Rac)-CP-601927 hydrochloride Structure
(Rac)-CP-601927 hydrochloride structure
Common Name (Rac)-CP-601927 hydrochloride
CAS Number 230615-01-7 Molecular Weight 263.69
Density N/A Boiling Point N/A
Molecular Formula C12H13ClF3N Melting Point N/A
MSDS N/A Flash Point N/A

 Use of (Rac)-CP-601927 hydrochloride


(Rac)-CP-601927 hydrochloride is the racemate of CP-601927. CP-601927 is a nAChR agonist with Ki values 1.2 nM and 102 nM for α4β2 and α3β4 nAChR, respectively[1].

 Names

Name (Rac)-CP-601927 hydrochloride

 (Rac)-CP-601927 hydrochloride Biological Activity

Description (Rac)-CP-601927 hydrochloride is the racemate of CP-601927. CP-601927 is a nAChR agonist with Ki values 1.2 nM and 102 nM for α4β2 and α3β4 nAChR, respectively[1].
Related Catalog
In Vitro CP-601927 induces significant antidepressant-like effects in mice. CP-601927 could decrease cholinergic signaling as a result of its reduced efficacy or via desensitization of α4β2* nAChRs[1].
References

[1]. Yann S Mineur, et al. α4β2 nicotinic acetylcholine receptor partial agonists with low intrinsic efficacy have antidepressant-like properties. Behav Pharmacol. 2011 Aug;22(4):291-9.

 Chemical & Physical Properties

Molecular Formula C12H13ClF3N
Molecular Weight 263.69
Top Suppliers:I want be here


Get all suppliers and price by the below link:

(Rac)-CP-601927 hydrochloride suppliers

(Rac)-CP-601927 hydrochloride price

Related Compounds: More...
CP-601927
357425-02-6
(Rac)-Verapamil D7 hydrochloride
1188265-55-5
PHENYL-2-AMINOPROPANE-1,1,2,3,3,3-D6 HCL
205437-60-1
rac Viloxazine-d5 Hydrochloride
117320-32-8
rac Methadone-d3 Hydrochloride
65566-72-5
rac-Soterenol-d7 Hydrochloride
14816-67-2
rac Tolterodine-d6 Hydrochloride
1330076-60-2
rac Rotigotine-d3 Hydrochloride Salt Also See R700703
1215846-20-0
(rac)-Metanephrine-d3 hydrochloride
1215507-88-2
5-(4-(dimethylamino)phenyl)-2-(isopentylthio)-7,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,5H)-dione
631853-45-7
2-(sec-butylthio)-5-phenyl-7,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,5H)-dione
631853-58-2
2-(butan-2-ylsulfanyl)-5-(4-methoxyphenyl)-5,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,7H)-dione
631853-72-0
2-(sec-butylthio)-5-(4-hydroxy-3-methoxyphenyl)-7,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,5H)-dione
631853-77-5
2-(sec-butylthio)-5-(thiophen-2-yl)-7,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,5H)-dione
631853-84-4
(R)-2-Amino-2-(2-chloro-6-iodophenyl)ethan-1-ol
1389361-97-0
2-(sec-butylthio)-5-(pyridin-4-yl)-7,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,5H)-dione
631853-89-9
2-(sec-butylthio)-5-(4-(dimethylamino)phenyl)-7,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,5H)-dione
631853-97-9
2-(butan-2-ylsulfanyl)-8,8-dimethyl-5-(thiophen-2-yl)-5,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,7H)-dione
631854-47-2
2-(sec-butylthio)-8,8-dimethyl-5-(5-methylfuran-2-yl)-7,8,9,10-tetrahydropyrimido[4,5-b]quinoline-4,6(3H,5H)-dione
631854-48-3