PROTAC VEGFR-2 degrader-2

Modify Date: 2025-11-13 23:06:25

PROTAC VEGFR-2 degrader-2 Structure
PROTAC VEGFR-2 degrader-2 structure
Common Name PROTAC VEGFR-2 degrader-2
CAS Number 2353417-85-1 Molecular Weight 930.10
Density N/A Boiling Point N/A
Molecular Formula C50H56FN9O6S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of PROTAC VEGFR-2 degrader-2


PROTAC VEGFR-2 degrader-2(PROTAC-4), a PROTAC VEGFR-2 degrader, exhibits little VEGFR-2 inhibition (IC50> 1 μM) and anti-proliferative activity against EA.hy926 cells (IC50> 100μM)[1].

 Names

Name PROTAC VEGFR-2 degrader-2

 PROTAC VEGFR-2 degrader-2 Biological Activity

Description PROTAC VEGFR-2 degrader-2(PROTAC-4), a PROTAC VEGFR-2 degrader, exhibits little VEGFR-2 inhibition (IC50> 1 μM) and anti-proliferative activity against EA.hy926 cells (IC50> 100μM)[1].
Related Catalog
References

[1]. Yuanyuan Shan, et al. Discovery of novel anti-angiogenesis agents. Part 11: Development of PROTACs based on active molecules with potency of promoting vascular normalization. Eur J Med Chem. 2020 Nov 1;205:112654.

 Chemical & Physical Properties

Molecular Formula C50H56FN9O6S
Molecular Weight 930.10
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