BET-IN-15

Modify Date: 2025-08-27 15:47:20

BET-IN-15 Structure
BET-IN-15 structure
Common Name BET-IN-15
CAS Number 2408994-22-7 Molecular Weight 444.45
Density N/A Boiling Point N/A
Molecular Formula C21H18F2N4O3S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of BET-IN-15


BET-IN-15 (compound 1) is a potent and orally active BET inhibitor with IC50 values of 0.64, 0.25 nM for BRD4-BD1, BRD4-BD2, respectively. BET-IN-15 shows antiproliferative activity[1].

 Names

Name BET-IN-15

 BET-IN-15 Biological Activity

Description BET-IN-15 (compound 1) is a potent and orally active BET inhibitor with IC50 values of 0.64, 0.25 nM for BRD4-BD1, BRD4-BD2, respectively. BET-IN-15 shows antiproliferative activity[1].
Related Catalog
Target

BRD4-BD1:0.64 nM (IC50)

BRD4-BD2:0.25 nM (IC50)

References

[1]. WenWei Xu, et al. Crystal form and salt form of bromine domain protein inhibitor and preparation method therefor. WO2021143922A1.

 Chemical & Physical Properties

Molecular Formula C21H18F2N4O3S
Molecular Weight 444.45
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