Sivopixant
Modify Date: 2024-01-03 11:51:46
Sivopixant structure
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Common Name | Sivopixant | ||
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| CAS Number | 2414285-40-6 | Molecular Weight | 507.93 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C25H22ClN5O5 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of SivopixantSivopixant (S-600918) is a potent and selective P2X3 receptor antagonist (P2X3 IC50=4.2 nM; P2X2/3 IC50=1100 nM). Sivopixant shows strong analgesic effect[1]. |
| Name | Sivopixant |
|---|
| Description | Sivopixant (S-600918) is a potent and selective P2X3 receptor antagonist (P2X3 IC50=4.2 nM; P2X2/3 IC50=1100 nM). Sivopixant shows strong analgesic effect[1]. |
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| Related Catalog | |
| In Vivo | Sivopixant (S-600918) (i.v.;1 mg/kg) shows a longer half-life (T1/2= 10.1 hours) and a strong analgesic effect in the rat Seltzer model of allodynia (ED50=0.4 mg/kg)[1]. |
| References |
| Molecular Formula | C25H22ClN5O5 |
|---|---|
| Molecular Weight | 507.93 |