EST73502 hydrochloride structure
|
Common Name | EST73502 hydrochloride | ||
---|---|---|---|---|
CAS Number | 2535970-65-9 | Molecular Weight | 388.88 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C19H27ClF2N2O2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of EST73502 hydrochlorideEST73502 hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 hydrochloride has antinociceptive activity. |
Name | EST73502 hydrochloride |
---|
Description | EST73502 hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 hydrochloride has antinociceptive activity. |
---|
Molecular Formula | C19H27ClF2N2O2 |
---|---|
Molecular Weight | 388.88 |