ARD-2051
Modify Date: 2024-01-13 16:47:50
ARD-2051 structure
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Common Name | ARD-2051 | ||
|---|---|---|---|---|
| CAS Number | 2632305-17-8 | Molecular Weight | 789.32 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C43H45ClN8O5 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of ARD-2051ARD-2051 is a potent and orally active androgen receptor (AR) proteolysis-targeting chimera degrader. ARD-2051 achieves DC50 values of 0.6 nM for AR protein degradation in both the LNCaP and VCaP prostate cancer cell lines. ARD-2051 can be used for the research of prostate cancer[1]. |
| Name | ARD-2051 |
|---|
| Description | ARD-2051 is a potent and orally active androgen receptor (AR) proteolysis-targeting chimera degrader. ARD-2051 achieves DC50 values of 0.6 nM for AR protein degradation in both the LNCaP and VCaP prostate cancer cell lines. ARD-2051 can be used for the research of prostate cancer[1]. |
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| Related Catalog | |
| Target |
DC50: 0.6 nM (AR protein degradation)[1] |
| References |
| Molecular Formula | C43H45ClN8O5 |
|---|---|
| Molecular Weight | 789.32 |