TAK-802 hydrochloride
Modify Date: 2024-04-02 11:33:45
TAK-802 hydrochloride structure
|
Common Name | TAK-802 hydrochloride | ||
|---|---|---|---|---|
| CAS Number | 263248-36-8 | Molecular Weight | 456.986 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C26H30ClFN2O2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of TAK-802 hydrochlorideA potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM; exhibits high selectivity for acetylcholinesterase inhibition over butyrylcholinesterase inhibition; increases rhythmic bladder contractions in Guinea pigs and rats without affecting the basal intravesical pressure. Other Indication Phase 2 Discontinued |
| Name | TAK-802 hydrochloride |
|---|
| Description | A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM; exhibits high selectivity for acetylcholinesterase inhibition over butyrylcholinesterase inhibition; increases rhythmic bladder contractions in Guinea pigs and rats without affecting the basal intravesical pressure. Other Indication Phase 2 Discontinued |
|---|---|
| References | References 1. Ishichi Y, et al. Bioorg Med Chem. 2005 Mar 15;13(6):1901-11. 2. Nagabukuro H, et al. Eur J Pharmacol. 2004 Feb 6;485(1-3):299-305. 3. Nagabukuro H, et al. Eur J Pharmacol. 2004 Jun 28;494(2-3):225-32. View Related Products by Target Acetylcholinesterase (AChE) Other Indication |
| Molecular Formula | C26H30ClFN2O2 |
|---|---|
| Molecular Weight | 456.986 |