Fesoterodine Fumarate structure
|
Common Name | Fesoterodine Fumarate | ||
---|---|---|---|---|
CAS Number | 286930-03-8 | Molecular Weight | 527.649 | |
Density | N/A | Boiling Point | 518.9ºC at 760 mmHg | |
Molecular Formula | C30H41NO7 | Melting Point | 72-78ºC | |
MSDS | N/A | Flash Point | 267.6ºC |
Use of Fesoterodine FumarateFesoterodine Fumarate is an antimuscarinic agent and is rapidly de-esterified to its active metabolite 5-hydroxymethyl tolterodine that is a muscarinic receptor antagonist.IC50 value:Target: mAChRFesoterodine has the advantage of allowing more flexible dosage than other muscarinic antagonists. Its tolerability and side effects are similar to other muscarinic antagonists and as a new drug seems unlikely to make great changes in practices of treatment for overactive bladder. |
Name | (E)-but-2-enedioic acid,[2-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-(hydroxymethyl)phenyl] 2-methylpropanoate |
---|---|
Synonym | More Synonyms |
Description | Fesoterodine Fumarate is an antimuscarinic agent and is rapidly de-esterified to its active metabolite 5-hydroxymethyl tolterodine that is a muscarinic receptor antagonist.IC50 value:Target: mAChRFesoterodine has the advantage of allowing more flexible dosage than other muscarinic antagonists. Its tolerability and side effects are similar to other muscarinic antagonists and as a new drug seems unlikely to make great changes in practices of treatment for overactive bladder. |
---|---|
Related Catalog | |
References |
[5]. Fesoterodine |
Boiling Point | 518.9ºC at 760 mmHg |
---|---|
Melting Point | 72-78ºC |
Molecular Formula | C30H41NO7 |
Molecular Weight | 527.649 |
Flash Point | 267.6ºC |
Exact Mass | 527.288330 |
PSA | 124.37000 |
LogP | 5.09290 |
Storage condition | Hygroscopic, Store under Inert atmosphere -20°C Freezer |
(R)-Fesoterodine fumarate |
Fesoterodine Fumarate |
UNII-EOS72165S7 |
SPM 8272 |
SPM 907 |
Propanoic acid, 2-methyl-, 2-[(1R)-3-[bis(1-methylethyl)amino]-1-phenylpropyl]-4-(hydroxymethyl)phenyl ester, (2E)-2-butenedioate (1:1) |
Toviaz,Fesoterodine fumarate |
2-[(1R)-3-(Diisopropylamino)-1-phenylpropyl]-4-(hydroxymethyl)phenyl 2-methylpropanoate (2E)-2-butenedioate (1:1) |
Propanoic acid,2-methyl-,2-((1R)-3-(bis(1-methylethyl)amino)-1-phenylpropyl)-4-(hydroxymethyl)phenyl ester,(2E)-2-butenedioate (1:1) (salt) |
Fesoterodinefumarate |
Toviaz |
(R)-2-(3-(Diisopropylamino)-1-phenylpropyl)-4-(hydroxymethyl)phenyl isobutyrate fumarate |
Fesoterodine (fumarate) |