MRS2298

Modify Date: 2024-01-28 22:26:02

MRS2298 Structure
MRS2298 structure
Common Name MRS2298
CAS Number 491611-43-9 Molecular Weight 431.66
Density 2.03±0.1 g/cm3(Predicted) Boiling Point 735.8±70.0 °C(Predicted)
Molecular Formula C10H16ClN5O8P2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of MRS2298


MRS2298? is a potent acyclic P2Y1 receptor antagonist with a Ki of 29.6 nM. MRS2298 inhibits the ADP-induced aggregation of human platelets with an IC50 of 62.8 nM. MRS2298 inhibits Ca2+ rise in platelets with an IC50 of 810 nM[1].

 Names

Name MRS2298
Synonym More Synonyms

 MRS2298 Biological Activity

Description MRS2298? is a potent acyclic P2Y1 receptor antagonist with a Ki of 29.6 nM. MRS2298 inhibits the ADP-induced aggregation of human platelets with an IC50 of 62.8 nM. MRS2298 inhibits Ca2+ rise in platelets with an IC50 of 810 nM[1].
Related Catalog
References

[1]. Marco Cattaneo, et al. Antiaggregatory activity in human platelets of potent antagonists of the P2Y 1 receptor. Biochem Pharmacol. 2004 Nov 15;68(10):1995-2002.  

 Chemical & Physical Properties

Density 2.03±0.1 g/cm3(Predicted)
Boiling Point 735.8±70.0 °C(Predicted)
Molecular Formula C10H16ClN5O8P2
Molecular Weight 431.66

 Synonyms

MRS 2298
MRS-2298