Clathrin-IN-4 structure
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Common Name | Clathrin-IN-4 | ||
|---|---|---|---|---|
| CAS Number | 762242-59-1 | Molecular Weight | 426.15 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C17H18Br2N2O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Clathrin-IN-4Clathrin-IN-4 (compound 8b), a Wiskostatin (HY-12534) analogue, is a potent inhibitor of clathrin mediated endocytosis with an IC50 of 2.1 μM. Clathrin-IN-4 is a dynamin I GTPase activity inhibitor with an IC50 of 9.1 μM[1]. |
| Name | Clathrin-IN-4 |
|---|
| Description | Clathrin-IN-4 (compound 8b), a Wiskostatin (HY-12534) analogue, is a potent inhibitor of clathrin mediated endocytosis with an IC50 of 2.1 μM. Clathrin-IN-4 is a dynamin I GTPase activity inhibitor with an IC50 of 9.1 μM[1]. |
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| Related Catalog | |
| References |
| Molecular Formula | C17H18Br2N2O |
|---|---|
| Molecular Weight | 426.15 |
| InChIKey | XUBJEDZHBUPBKL-CYBMUJFWSA-N |
| SMILES | CN(C)CC(O)Cn1c2ccc(Br)cc2c2cc(Br)ccc21 |
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Source: ChEMBL
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External Id: CHEMBL4513082
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Source: ChEMBL
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Name: Inhibition of phosphotidylserine liposome-stimulated Dynamin 1 (unknown origin) GTPas...
Source: ChEMBL
Target: Dynamin-1
External Id: CHEMBL5356087
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Name: Inhibition of clathrin-mediated endocytosis in serum-starved human U2OS cells assesse...
Source: ChEMBL
Target: N/A
External Id: CHEMBL5356088
|