δ-Endorphin (human) structure
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Common Name | δ-Endorphin (human) | ||
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CAS Number | 76622-84-9 | Molecular Weight | 3022.47 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C139H217N33O40S | Melting Point | N/A | |
MSDS | USA | Flash Point | N/A |
Use of δ-Endorphin (human)β-Endorphin (1-27) (human) is an opioid antagonist that binds μ-, δ-, and κ-opioid receptors with Kis of 5.31, 6.17, and 39.82 nM, respectively. β-Endorphin (1-27) (human) inhibits β-Endorphin (HY-P1502)-induced and etorphine-induced analgesia[1][2]. |
Name | δ-Endorphin (human) |
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Synonym | More Synonyms |
Description | β-Endorphin (1-27) (human) is an opioid antagonist that binds μ-, δ-, and κ-opioid receptors with Kis of 5.31, 6.17, and 39.82 nM, respectively. β-Endorphin (1-27) (human) inhibits β-Endorphin (HY-P1502)-induced and etorphine-induced analgesia[1][2]. |
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Related Catalog | |
Target |
Ki: 5.31 nM (μ-opioid receptor), 6.17 nM (δ-opioid receptor), 39.82 nM (κ-opioid receptor)[1] |
References |
Molecular Formula | C139H217N33O40S |
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Molecular Weight | 3022.47 |
Exact Mass | 3020.57000 |
PSA | 1222.67000 |
LogP | 3.79500 |
Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
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RIDADR | NONH for all modes of transport |
WGK Germany | 3 |
beta-Endorphin huMan fragMent 1-27 |
5-[[5-amino-1-[[2-[[4-amino-1-[[1-[2-[[1-[[1-[[1-[[1-[[2-[[5-amino-1-[[3-amino-1-[[2-[[1-[[1-[[5-amino-1-[[3-amino-1-[[2-[[1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-methyl-2-oxo-ethyl]carbamoyl]-3-oxo-propyl]carbamoyl]pentyl]carbamoyl]-2-methyl-butyl]carbamoyl]-2-methyl-butyl]amino]-1-methyl-2-oxo-ethyl]carbamoyl]-3-oxo-propyl]carbamoyl]pentyl]amino]-1-benzyl-2-oxo-ethyl]carbamoyl]-3-methyl-butyl]carbamoyl]-2-hydroxy-propyl]carbamoyl]-2-methyl-propyl]carbamoyl]-3-methyl-butyl]carbamoyl]pyrrolidine-1-carbonyl]-2-hydroxy-propyl]carbamoyl]-4-oxo-butyl]amino]-1-(hydroxymethyl)-2-oxo-ethyl]carbamoyl]pentyl]amino]-4-[[2-[[2-[[2-[[2-[[2-[[2-[[2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenyl-propanoyl]amino]-4-methylsulfanyl-butanoyl]amino]-3-hydroxy-butanoyl]amino]-3-hydroxy-propanoyl]amino]-5-oxo-pentanoic acid |