LAS101057 structure
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Common Name | LAS101057 | ||
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CAS Number | 925676-48-8 | Molecular Weight | 335.33500 | |
Density | 1.400±0.06 g/cm3 (20 °C, 760 mmHg) | Boiling Point | 509.2±50.0 °C (760 mmHg) | |
Molecular Formula | C18H14FN5O | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of LAS101057LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. |
Name | Cyclopropanecarboxamide, N-[5-(3-fluoro-4-pyridinyl)-6-(3-pyridinyl)-2-pyrazinyl] |
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Synonym | More Synonyms |
Description | LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. |
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Related Catalog | |
In Vivo | At 3 mg/kg, LAS101057 is active in preventing methacholine-induced AHR, and at 10 mg/kg it inhibits AHR to methacholine to a level virtually equal to that seen with dexamethasone at 1 mg/kg[1]. |
References |
Density | 1.400±0.06 g/cm3 (20 °C, 760 mmHg) |
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Boiling Point | 509.2±50.0 °C (760 mmHg) |
Molecular Formula | C18H14FN5O |
Molecular Weight | 335.33500 |
Exact Mass | 335.11800 |
PSA | 80.66000 |
LogP | 3.16120 |
las-101057 |
LAS101057 |