Tetrahedron letters

Direct palladium-catalyzed C-3 arylation of indoles

Z Zhang, Z Hu, Z Yu, P Lei, H Chi, Y Wang, R He

Index: Zhang, Zhiqiang; Hu, Zhizhi; Yu, Zhixiao; Lei, Peng; Chi, Haijun; Wang, Yue; He, Ren Tetrahedron Letters, 2007 , vol. 48, # 13 p. 2415 - 2419

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Citation Number: 77

Abstract

Indole derivatives are one of the most important and commonly found heterocyclic motifs in both pharmaceuticals and natural products, 1 since indole can be considered as a commonly used starting material for further alkaloid synthesis if suitable synthetic methodology can be developed from this parent skeleton. 2 The Pd-catalyzed arylation of indole is a quite hot research area in recent years. In most cases, this type of Pd-catalyzed reaction gave 2-arylated indole 3 ...

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