Synthesis

Efficient synthesis of 1, 5-disubstituted tetrazoles

AR Katritzky, C Cai, NK Meher

Index: Katritzky, Alan R.; Cai, Chunming; Meher, Nabin K. Synthesis, 2007 , # 8 p. 1204 - 1208

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Citation Number: 37

Abstract

However, many of these reported methods suffer from one or more of the following drawbacks: (i) long reaction times, (ii) the use of toxic and/or explosive reagents, (iii) tedious workup and low yields, (iv) high temperatures, (v) the formation of inseparable regioisomers, and (vi) the use of uncommon starting materials. Thus, a mild and efficient method is required for the preparation of 1,5-disubstituted tetrazoles. ... Imidoylbenzotriazoles, which are ...

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