Dynamic kinetic asymmetric transformation of diene monoepoxides: A practical asymmetric synthesis of vinylglycinol, vigabatrin, and ethambutol

BM Trost, RC Bunt, RC Lemoine…

Index: Journal of the American Chemical Society, , vol. 122, # 25 p. 5968 - 5976

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Citation Number: 205

Abstract

... Journal of ... Chem. Soc. , 2000, 122 (25), pp 5968–5976. DOI: 10.1021/ja000547d. Publication Date (Web): June 8, 2000. Copyright © 2000 American Chemical Society. ... 5 The utility of vinylglycinol as a chiral building block 6 led us to focus on phthalimide as the pro-nucleophile. ...

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