Tetrahedron

2-Amino-6-iodo-4-tosyloxypyrimidine: a versatile key intermediate for regioselective functionalization of 2-aminopyrimidines in 4-and 6-positions

P Benderitter, JX de Araújo Júnior, M Schmitt…

Index: Benderitter, Pascal; de Araujo Junior, Joao Xavier; Schmitt, Martine; Bourguignon, Jean-Jacques Tetrahedron, 2007 , vol. 63, # 50 p. 12465 - 12470

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Citation Number: 16

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... 2-Amino-6-iodo-4-tosyloxypyrimidine, easily prepared from commercially available material, is a key intermediate for the preparation of differentially substituted 2-aminopyrimidines by means of sequenced Suzuki and/or Sonogashira reactions. ... Examples of 2-aminopyrimidines ...

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