Rh-catalyzed intramolecular debenzylative cyclization of amines. Butyrolactams from benzylamines having a chloroacetylene moiety
YT Oh, K Senda, T Hata, H Urabe
Index: Oh, Yun Taek; Senda, Kousuke; Hata, Takeshi; Urabe, Hirokazu Tetrahedron Letters, 2011 , vol. 52, # 19 p. 2458 - 2461
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Citation Number: 6
Abstract
Abstract When benzylamines having a chloroacetylene moiety were heated in wet toluene with a catalytic amount of rhodium trifluoroacetate dimer, intramolecular debenzylative cyclization took place to give butyrolactams. This method is a new entry to selective debenzylation of amines.
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