3-Oxo-N-phenylbutanamide

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Names

[ CAS No. ]:
102-01-2

[ Name ]:
3-Oxo-N-phenylbutanamide

[Synonym ]:
acetoacetamidobenzene
Linazol
Coupler 633
Acetoacetanilide
a-Acetylacetanilide
usafek-1239
2-acetylacetanilide
Acetoacetanilid
MFCD00008780
1V1VMR
N-(Acetylacetyl)aniline
N-Phenyl-3-ketobutanamide
AAA
Cetoactanilide
EINECS 202-996-4
(1E)-3-Oxo-N-phenylbutanimidic acid
b-Ketobutyranilide
acetoacetylaminobenzene
3-Oxo-N-phenylbutanamide
Butanamide, 3-oxo-N-phenyl-
Butanimidic acid, 3-oxo-N-phenyl-, (1E)-
acetoacetic anilide
AAN
acetoacetyl-phenylamine
Acetoacetonilide
1-(N-phenylcarbamyl)propan-2-one

Chemical & Physical Properties

[ Density]:
1.1±0.1 g/cm3

[ Boiling Point ]:
329.0±44.0 °C at 760 mmHg

[ Melting Point ]:
83-88 °C(lit.)

[ Molecular Formula ]:
C10H11NO2

[ Molecular Weight ]:
177.200

[ Flash Point ]:
152.8±28.4 °C

[ Exact Mass ]:
177.078979

[ PSA ]:
46.17000

[ LogP ]:
1.43

[ Vapour density ]:
6.1 (vs air)

[ Vapour Pressure ]:
0.0±0.8 mmHg at 25°C

[ Index of Refraction ]:
1.532

[ Stability ]:
Stable. Combustible. Incompatible with strong oxidizing agents.

[ Water Solubility ]:
5 g/L (20 ºC)

MSDS

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
AK4200000
CHEMICAL NAME :
Acetoacetanilide
CAS REGISTRY NUMBER :
102-01-2
LAST UPDATED :
199806
DATA ITEMS CITED :
15
MOLECULAR FORMULA :
C10-H11-N-O2
MOLECULAR WEIGHT :
177.22
WISWESSER LINE NOTATION :
1V1VMR

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
2450 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0533750
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
800 mg/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Vascular - regional or general arteriolar or venous dilation Lungs, Thorax, or Respiration - cyanosis
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0533572
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Subcutaneous
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
7 gm/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
GTPZAB Gigiena Truda i Professional'nye Zabolevaniya. Labor Hygiene and Occupational Diseases. (V/O Mezhdunarodnaya Kniga, 113095 Moscow, USSR) V.1-36, 1957-1992. For publisher information, see MTPEEI Volume(issue)/page/year: 31(1),49,1987
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
3400 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
GTPZAB Gigiena Truda i Professional'nye Zabolevaniya. Labor Hygiene and Occupational Diseases. (V/O Mezhdunarodnaya Kniga, 113095 Moscow, USSR) V.1-36, 1957-1992. For publisher information, see MTPEEI Volume(issue)/page/year: 31(1),49,1987
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
300 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: AD277-689
TYPE OF TEST :
LDLo - Lowest published lethal dose
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Mammal - cat
DOSE/DURATION :
500 mg/kg
TOXIC EFFECTS :
Blood - methemoglobinemia-carboxyhemoglobin
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0534808-1
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rabbit
DOSE/DURATION :
3925 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
GTPZAB Gigiena Truda i Professional'nye Zabolevaniya. Labor Hygiene and Occupational Diseases. (V/O Mezhdunarodnaya Kniga, 113095 Moscow, USSR) V.1-36, 1957-1992. For publisher information, see MTPEEI Volume(issue)/page/year: 31(1),49,1987
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Administration onto the skin
SPECIES OBSERVED :
Rodent - guinea pig
DOSE/DURATION :
>1 gm/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0533572 ** OTHER MULTIPLE DOSE TOXICITY DATA **
TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
14024 mg/kg/14D-C
TOXIC EFFECTS :
Sense Organs and Special Senses (Eye) - effect, not otherwise specified Blood - changes in erythrocyte (RBC) count Nutritional and Gross Metabolic - weight loss or decreased weight gain
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0533572 *** OCCUPATIONAL EXPOSURE LIMITS *** OEL-RUSSIA:STEL 1 mg/m3;Skin JAN 1993 *** NIOSH STANDARDS DEVELOPMENT AND SURVEILLANCE DATA *** NIOSH OCCUPATIONAL EXPOSURE SURVEY DATA : NOHS - National Occupational Hazard Survey (1974) NOHS Hazard Code - 84311 No. of Facilities: 53 (estimated) No. of Industries: 2 No. of Occupations: 3 No. of Employees: 1062 (estimated) NOES - National Occupational Exposure Survey (1983) NOES Hazard Code - 84311 No. of Facilities: 50 (estimated) No. of Industries: 1 No. of Occupations: 3 No. of Employees: 1108 (estimated)

Safety Information

[ Symbol ]:

GHS07

[ Signal Word ]:
Warning

[ Hazard Statements ]:
H302-H312

[ Precautionary Statements ]:
P280

[ Personal Protective Equipment ]:
dust mask type N95 (US);Eyeshields;Gloves

[ Hazard Codes ]:
Xn:Harmful

[ Risk Phrases ]:
R21/22

[ Safety Phrases ]:
S36

[ RIDADR ]:
NONH for all modes of transport

[ WGK Germany ]:
1

[ RTECS ]:
AK4200000

[ HS Code ]:
2924299090

Synthetic Route

Precursor & DownStream

Precursor

  • tert-Butyl acetoacetate
  • Methyl acetoacetate
  • 2,2,6-Trimethyl-4H-1,3-dioxin-4-one
  • Ethyl acetoacetate
  • DIAZOACETONE
  • carbon monoxide

DownStream

  • 1,1,3,3-Tetrabutylurea
  • Urea,N,N-dibutyl-N'-phenyl-
  • 2-chloro-3-oxo-n-phenylbutanamide
  • 2,4-dimethyl-6-oxo-N,1-diphenylpyridine-3-carboxamide
  • 4-methylquinolin-2-ol
  • ethyl 4-methyl-2-oxoquinoline-1-carboxylate
  • 2-[bis(methylsulfanyl)methylidene]-3-oxo-N-phenylbutanamide
  • 3-Methyl-3-pyrazolin-5-one
  • 4-oxo-N-phenylpentanamide

Customs

[ HS Code ]: 2924299090

[ Summary ]:
2924299090. other cyclic amides (including cyclic carbamates) and their derivatives; salts thereof. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:30.0%

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Related Compounds

  • 3-oxo-N-phenylbutanamide
  • 3-oxo-n-phenylbutanamide
  • 4-Bromo-3-oxo-N-phenylbutanamide
  • 2-ethyl-3-oxo-N-phenylbutanamide
  • N-ethyl-3-oxo-N-phenylbutanamide
  • 2-benzyl-3-oxo-N-phenylbutanamide
  • Methyl 2-methyl-4-(methylsulfonyl)pyrimidine-5-carboxylate
  • 5-Bromo-3-methylpyrazolo[1,5-a]pyrimidine
  • tert-Butyl 4-amino-2-cyanobenzoate
  • tert-Butyl 3-formylpicolinate
  • tert-Butyl (2-(4-iodophenyl)propan-2-yl)carbamate
  • tert-Butyl (cyano(piperidin-2-yl)methyl)carbamate
  • (R)-1-(5-Chloro-2-fluoropyridin-3-yl)ethanol
  • tert-Butyl 2-amino-5-(2-fluorophenyl)thiazole-4-carboxylate
  • tert-Butyl ((4-bromopyridin-2-yl)methyl)(methyl)carbamate
  • Isopropyl 6-(hydroxymethyl)picolinate