CGP 20712 A

Suppliers

Names

[ CAS No. ]:
105737-62-0

[ Name ]:
CGP 20712 A

[Synonym ]:
2-hydroxy-5-[2-[[2-hydroxy-3-[4-[1-methyl-4-(trifluoromethyl)imidazol-2-yl]phenoxy]propyl]amino]ethoxy]benzamide,methanesulfonic acid

Chemical & Physical Properties

[ Boiling Point ]:
764.8ºC at 760mmHg

[ Molecular Formula ]:
C24H29F3N4O8S

[ Molecular Weight ]:
590.56900

[ Flash Point ]:
416.3ºC

[ Exact Mass ]:
590.16600

[ PSA ]:
194.61000

[ LogP ]:
3.99470

[ Vapour Pressure ]:
9.69E-23mmHg at 25°C

[ Storage condition ]:
2-8°C

MSDS

Safety Information

[ Personal Protective Equipment ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ RIDADR ]:
NONH for all modes of transport

[ WGK Germany ]:
3

Articles

CGP 20712 A: a useful tool for quantitating beta 1- and beta 2-adrenoceptors.

Eur. J. Pharmacol. 130 , 137-139, (1986)

CGP 20712 A (1-[2-((3-carbamoyl-4-hydroxy)phenoxy)ethylamino]-3- [4-(1-methyl-4-trifluoromethyl-2-imidazolyl) phenoxy]-2-propanol methanesulfonate), a specific beta 1-adrenoceptor antagonist, was test...

Beta-adrenoceptor subtypes in human coronary artery: desensitization of beta 2-adrenergic vasorelaxation by chronic beta 1-adrenergic stimulation in vitro.

J. Cardiovasc. Pharmacol. 25 , 134-141, (1995)

We previously demonstrated that right atrial strips from patients treated with beta 1-selective antagonists exhibit sensitization of beta 2-adrenergic responses in vitro. We also showed that cardiac b...


More Articles


Related Compounds

  • CGP 20712 dihydrochloride
  • 1-[2-((3-carbamoyl-4-hydroxy)phenoxy)ethylamino]-3-[4-(1-methyl-4-trifluoromethyl-2-imidazolyl)phenoxy]propan-2-ol
  • CGP 3466B maleate
  • cgp 46251
  • Formoterol Hemifumarate
  • Sercloremine hydrochloride