Pipazethate

Suppliers

Names

[ CAS No. ]:
2167-85-3

[ Name ]:
Pipazethate

[Synonym ]:
4-Aza-phenothiazin-10-carbonsaeure-piperidino-aethoxy-aethylester
Pipazetato [INN-Spanish]
Pipazetate
Pipazetatum [INN-Latin]
pipazethate
Theratuss
benzo[b]pyrido[2,3-e][1,4]thiazine-10-carboxylic acid 2-(2-piperidin-1-yl-ethoxy)-ethyl ester
Lenopect

Chemical & Physical Properties

[ Density]:
1.26g/cm3

[ Boiling Point ]:
553.3ºC at 760mmHg

[ Molecular Formula ]:
C21H25N3O3S

[ Molecular Weight ]:
399.50700

[ Flash Point ]:
288.4ºC

[ Exact Mass ]:
399.16200

[ PSA ]:
80.20000

[ LogP ]:
4.32630

[ Vapour Pressure ]:
2.76E-12mmHg at 25°C

[ Index of Refraction ]:
1.612

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
UU8485000
CHEMICAL NAME :
10H-Pyrido(3,2-b)(1,4)benzothiazine-10-carboxylic acid, 2-(2-(1-piperidinyl)ethoxy) ethyl ester
CAS REGISTRY NUMBER :
2167-85-3
LAST UPDATED :
199612
DATA ITEMS CITED :
2
MOLECULAR FORMULA :
C21-H25-N3-O3-S
MOLECULAR WEIGHT :
399.55

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
94647 ug/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
AIPTAK Archives Internationales de Pharmacodynamie et de Therapie. (Heymans Institute of Pharmacology, De Pintelaan 185, B-9000 Ghent, Belgium) V.4- 1898- Volume(issue)/page/year: 188,189,1970
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
13140 ug/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
AIPTAK Archives Internationales de Pharmacodynamie et de Therapie. (Heymans Institute of Pharmacology, De Pintelaan 185, B-9000 Ghent, Belgium) V.4- 1898- Volume(issue)/page/year: 188,189,1970

Synthetic Route

Click to get detail synthetic route

Precursor & DownStream

Precursor

  • 1H-Pyrido[3,2-b][1,4]benzothiazine
  • 2-(2-(Piperidyl)ethoxy)ethanol
  • 10H-pyrido[3,2-b][1,4]benzothiazine-10-carbonyl chloride

DownStream

Related Compounds

  • pipazethate
  • Pipazethate hydrochloride
  • N-(1,1-dioxidotetrahydro-3-thienyl)-2-(5-methyl-7-oxo-3-phenyl-7H-furo[3,2-g]chromen-6-yl)acetamide
  • N~1~-(1,3-benzothiazol-2-yl)-3-(3,5-dimethyl-7-oxo-7H-furo[3,2-g]chromen-6-yl)propanamide
  • 6-(Trimethylsilyl)-6-undecanol
  • 2-[(1-Ethylindol-3-yl)methylene]-3-oxobenzo[3,4-b]furan-6-yl 2-bromobenzoate
  • (3,4-Dichlorophenyl)methanesulfonyl fluoride
  • (4-Fluorophenyl)methanesulfonyl fluoride
  • N-methyl-4-oxopentanamide
  • 2-[4-(2-fluorophenyl)piperazin-1-yl]-N-(5-oxo-5,6,7,8-tetrahydroquinazolin-2-yl)acetamide
  • (2E)-3-(2,4,6-trimethylphenyl)prop-2-en-1-ol
  • 5-(4-bromophenyl)-N-[5-methoxy-2-(4-morpholinyl)phenyl]-2-furamide
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