Berberine hydrochloride

Suppliers

Names

[ CAS No. ]:
633-65-8

[ Name ]:
Berberine hydrochloride

[Synonym ]:
1,3-Benzodioxolo[5,6-a]benzo[g]quinolizinium, 5,6-dihydro-9,10-dimethoxy-, hydrochloride (1:1)
EINECS 211-195-9
berberine hydrochloride
BERBERINE HCL
5,6-dihydro-9,10-dimethoxy-1,3-benzodioxolo[5,6-a]benzo[g]quinolizinium chloride (1:1)
MFCD00011939
9,10-dimethoxy-5,6-dihydro[1,3]dioxolo[4,5-g]isoquino[3,2-a]isoquinolin-7-ium chloride
Berberine (chloride)

Chemical & Physical Properties

[ Density]:
1.654g/cm3

[ Melting Point ]:
200ºC

[ Molecular Formula ]:
C20H18ClNO4

[ Molecular Weight ]:
372.822

[ Exact Mass ]:
372.099701

[ PSA ]:
40.80000

[ LogP ]:
0.10030

[ Water Solubility ]:
SOLUBLE IN COLD WATER

MSDS

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
DR9866400
CHEMICAL NAME :
Berbinium, 7,8,13,13a-tetradehydro-9,10-dimethoxy-2,3-(methylene dioxy)-, chloride
CAS REGISTRY NUMBER :
633-65-8
LAST UPDATED :
199701
DATA ITEMS CITED :
9
MOLECULAR FORMULA :
C20-H18-N-O4.Cl
MOLECULAR WEIGHT :
371.84

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
>15 gm/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Nutritional and Gross Metabolic - body temperature decrease
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
60 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
>29586 mg/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Nutritional and Gross Metabolic - body temperature decrease
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
37 mg/kg
TOXIC EFFECTS :
Behavioral - convulsions or effect on seizure threshold Behavioral - excitement Lungs, Thorax, or Respiration - dyspnea
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Unreported
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
30 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value

MUTATION DATA

TYPE OF TEST :
DNA damage
TEST SYSTEM :
Mammal - species unspecified Lymphocyte
DOSE/DURATION :
22 umol/L
REFERENCE :
IJBBBQ Indian Journal of Biochemistry and Biophysics. (Publications & Information Directorate, CSIR, Hillside Rd., New Delhi 110 012, India) V.8- 1971- Volume(issue)/page/year: 18,245,1981

Safety Information

[ Personal Protective Equipment ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ Hazard Codes ]:
Xn: Harmful;

[ Risk Phrases ]:
R20/21/22

[ Safety Phrases ]:
S24/25

[ RIDADR ]:
UN 1544

[ WGK Germany ]:
2

[ RTECS ]:
DR9866400

[ Packaging Group ]:
III

[ Hazard Class ]:
6.1(b)

[ HS Code ]:
3003409000

Synthetic Route

Precursor & DownStream

Precursor

  • Dihydroberberine

DownStream

  • Dihydroberberine
  • Pyrimido[4,5-g]quinazoline-4,9-dione,3,8-dihydro-5,10-dihydroxy-2,7-bis(hydroxymethyl)-3,8-dimethyl-
  • Allocryptopine
  • Berberine
  • Coptisine chloride
  • Tetrahydroberberine
  • Berberrubine
  • Demethyleneberberine
  • Berberinol
  • 8-Oxyberberine

Customs

[ HS Code ]: 3003409000

Articles

Berberine blocks the relapse of Clostridium difficile infection in C57BL/6 mice after standard vancomycin treatment.

Antimicrob. Agents Chemother. 59 , 3726-35, (2015)

Vancomycin is a preferred antibiotic for treating Clostridium difficile infection (CDI) and has been associated with a rate of recurrence of CDI of as high as 20% in treated patients. Recent studies h...

Functional cloning and characterization of the multidrug efflux pumps NorM from Neisseria gonorrhoeae and YdhE from Escherichia coli.

Antimicrob. Agents Chemother. 52 , 3052-60, (2008)

Active efflux of antimicrobial agents is one of the most important adapted strategies that bacteria use to defend against antimicrobial factors that are present in their environment. The NorM protein ...

Synergistic topical application of salt-processed Phellodendron amurense and Sanguisorba officinalis Linne alleviates atopic dermatitis symptoms by reducing levels of immunoglobulin E and pro-inflammatory cytokines in NC/Nga mice.

Mol. Med. Report. 12 , 7657-64, (2015)

Atopic dermatitis is a chronic inflammatory skin disease, and salt-processed Phellodendron amurense (CPE) and Sanguisorba officinalis Linne (SOE) are widely used as anti-inflammatory agents in Asia. T...


More Articles


Related Compounds

  • berberine hydrochloride hydrate
  • Berberine hydrochloride bihydrate
  • Berberine ursodeoxycholate
  • Berberine (chloride hydrate)
  • carnitine hydrochloride
  • Triprolidine hydrochloride
  • 2-(5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrol-2-yl)-3-(trifluoromethyl)pyridine
  • 9-(2-methoxyethyl)-6-{5-[2-(trifluoromethyl)pyridin-4-yl]-octahydropyrrolo[3,4-c]pyrrol-2-yl}-9H-purine
  • 4-Phenyl-1-[4-(trifluoromethyl)pyridin-2-yl]piperidine-4-carbonitrile
  • N-[(2,6-difluorophenyl)methyl]-6-(3,5-dimethyl-1H-pyrazol-1-yl)pyrimidin-4-amine
  • N-tert-butyl-4-[6-(pyrimidin-5-yl)-1,8-naphthyridin-2-yl]piperidine-1-carboxamide
  • 6-[5-(5-ethylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-9-(2-methoxyethyl)-9H-purine
  • 4-({4-[9-(2-methoxyethyl)-9H-purin-6-yl]piperazin-1-yl}methyl)benzonitrile
  • 5-fluoro-N,6-dimethyl-N-{[1-(3-methylquinoxalin-2-yl)piperidin-4-yl]methyl}pyrimidin-4-amine
  • N-[1-(1H-1,3-benzodiazol-2-yl)piperidin-3-yl]-N,5-dimethylpyrimidin-2-amine
  • N-[1-(4-methanesulfonyl-1,3-benzothiazol-2-yl)piperidin-3-yl]-N,5-dimethylpyrimidin-2-amine
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