Ethyl 2-Chloroacetoacetate

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Names

[ CAS No. ]:
638-07-3

[ Name ]:
Ethyl 2-Chloroacetoacetate

[Synonym ]:
4-chloro ethyl acetoacetate
Ethyl4-chloroacetoacetate
Ethyl (chloroacetyl)acetate
Butanoic acid, 4-chloro-3-oxo-, ethyl ester
Butanoic acid, 4-chloro-3-oxo-ethylester
Ethyl g-chloroacetoacetate
Ethyl-4-chloracetoacetat
Ethyl 4-chloroacetoa
Ethyl 4-chloro-3-oxobutyrate
4-Chloro-acetoacetic
ethyl 2-chloro-acetoacetate
Ethyl 4-chloro-3-oxobutanoate
MFCD00000939
Ethyl-4chloroacetaacetate
Ethyl 2-Chloroacetoacetate
Ethyl α-chloroacetoacetate
2-Chloroacetoacetic acid ethyl ester
Ethyl 4-chloroacetoacetate
EINECS 211-317-0

Chemical & Physical Properties

[ Density]:
1.2±0.1 g/cm3

[ Boiling Point ]:
235.5±0.0 °C at 760 mmHg

[ Melting Point ]:
-8 °C

[ Molecular Formula ]:
C6H9ClO3

[ Molecular Weight ]:
164.587

[ Flash Point ]:
96.7±0.0 °C

[ Exact Mass ]:
164.024017

[ PSA ]:
43.37000

[ LogP ]:
1.54

[ Vapour Pressure ]:
0.1±0.4 mmHg at 25°C

[ Index of Refraction ]:
1.436

[ Storage condition ]:
2-8°C

[ Water Solubility ]:
47.5 g/L (20 ºC)

MSDS

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
AK5110000
CHEMICAL NAME :
Acetoacetic acid, 4-chloro-, ethyl ester
CAS REGISTRY NUMBER :
638-07-3
BEILSTEIN REFERENCE NO. :
1761275
LAST UPDATED :
199710
DATA ITEMS CITED :
7
MOLECULAR FORMULA :
C6-H9-Cl-O3

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
200 mg/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Behavioral - tremor Skin and Appendages - hair
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0555360
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
108 mg/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Behavioral - convulsions or effect on seizure threshold Lungs, Thorax, or Respiration - respiratory depression
REFERENCE :
OYYAA2 Oyo Yakuri. Pharmacometrics. (Oyo Yakuri Kenkyukai, CPO Box 180, Sendai 980-91, Japan) V.1- 1967- Volume(issue)/page/year: 33,695,1987
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
150 mg/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Behavioral - tremor Skin and Appendages - hair
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0555360
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
88 mg/kg
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Behavioral - convulsions or effect on seizure threshold Lungs, Thorax, or Respiration - respiratory depression
REFERENCE :
OYYAA2 Oyo Yakuri. Pharmacometrics. (Oyo Yakuri Kenkyukai, CPO Box 180, Sendai 980-91, Japan) V.1- 1967- Volume(issue)/page/year: 33,695,1987 ** OTHER MULTIPLE DOSE TOXICITY DATA **
TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
750 mg/kg/15D-I
TOXIC EFFECTS :
Gastrointestinal - gastritis Gastrointestinal - ulceration or bleeding from stomach Liver - other changes
REFERENCE :
NTIS** National Technical Information Service. (Springfield, VA 22161) Formerly U.S. Clearinghouse for Scientific & Technical Information. Volume(issue)/page/year: OTS0555360

Safety Information

[ Symbol ]:

GHS05, GHS06

[ Signal Word ]:
Danger

[ Hazard Statements ]:
H301-H314

[ Precautionary Statements ]:
P280-P301 + P310-P305 + P351 + P338-P310

[ Personal Protective Equipment ]:
Faceshields;full-face respirator (US);Gloves;Goggles;multi-purpose combination respirator cartridge (US);type ABEK (EN14387) respirator filter

[ Hazard Codes ]:
T:Toxic;N:Dangerousfortheenvironment;

[ Risk Phrases ]:
R24/25;R34;R51/53

[ Safety Phrases ]:
S26-S36-S45-S61-S36/37/39

[ RIDADR ]:
UN 2922 8/PG 2

[ WGK Germany ]:
3

[ RTECS ]:
AK5110000

[ Packaging Group ]:
II

[ Hazard Class ]:
8

[ HS Code ]:
2918990090

Synthetic Route

Precursor & DownStream

Precursor

  • ETHYL 4,4-DICHLORO-3-OXOBUTANOATE
  • 4-chloro-3-oxobutanoyl chloride
  • Ethanol
  • 2-Hexanone
  • Benzaldehyde

DownStream

  • (3-ETHOXYCARBONYL-2-OXOPROPLY)TRIPHENYLPHOSPHONIUM CHLORIDE
  • diethyl 2-(chloromethyl)-6-methyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate
  • ETHYL 2-HYDROXY-5-METHYLBENZOATE
  • Hydrazinecarbothioamide,N-(4-methoxyphenyl)-
  • Diethyl succinosuccinate
  • ETHANONE, 1-(5-BROMO-2-BENZOFURANYL)-
  • octyl 4-chloro-3-oxobutanoate
  • Ethyl (6-chloroimidazo[1,2-a]pyridin-2-yl)acetate
  • 2-acetyl-7-methoxybenzofuran

Customs

[ HS Code ]: 2918300090

[ Summary ]:
2918300090 other carboxylic acids with aldehyde or ketone function but without other oxygen function, their anhydrides, halides, peroxides, peroxyacids and their derivatives。Supervision conditions:None。VAT:17.0%。Tax rebate rate:9.0%。MFN tariff:6.5%。General tariff:30.0%

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Related Compounds

  • Ethyl 2-Chloroacetoacetate
  • ethyl 2-amino-2-prop-2-ynylpent-4-ynoate
  • ethyl 2-(3,4-dichlorophenyl)sulfanylacetate
  • ethyl 2-[(N-hexylanilino)methyl]benzoate
  • ethyl 2-cyanohept-6-enoate
  • ethyl 2-(pyrrolidin-1-ylamino)cyclopentene-1-carboxylate
  • 4-((Cyclohexylamino)methyl)benzoic acid hydrochloride
  • 1-[(2,4-Dichlorophenyl)methyl]-N-(1,1-dimethylethyl)-2-methyl-1H-indole-3-methanamine
  • 2-Methoxy-6-(pyrazol-1-yl)-benzonitrile
  • 6-Ethoxy-N-(thietan-3-yl)pyridin-2-amine
  • m-Phenylenediamine-15n
  • 2-(2-Methoxy-7,8-dihydro-1H-benzofuro[4,5-d]imidazol-1-yl)ethan-1-amine
  • N-[(2-Methyl-1,3-dihydroisoindol-1-yl)methyl]prop-2-enamide
  • 2-Amino-1-(4-methylfuran-3-yl)propan-1-one
  • 2-(2,2-Difluoroethenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane
  • 1H-3-Benzazepin-7-ol, 8-chloro-2,3,4,5-tetrahydro-5-(3-iodophenyl)-3-methyl-, (S)-