| 常用名 | PF-04577806 | CAS号 | 1072100-81-2 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: PF-04577806 is a potent, selective and ATP competitive PKC inhibitor. PF-04577806 shows potent inhibitory activity towards PKCα, PKCβI, PKCβII, PKCγ, and PKCθ with IC50s of 2.4 nM, 8.1 nM, 6.9 nM, 45.9 nM, and 29.5 nM, respectively. PF-04577806 can reverse retinal vascular leakage in diabetic rats[1]. 物理化学性质: CAS号:1072100-81-2 常用中文名:PF-04577806 常用英文名:PF-04577806 分子式:C26H37N7O3 分子量:495.62 密度:1.2±0.1 g/cm3 沸点:613.4±55.0 °C at 760 mmHg 熔点:N/A 闪点:324.8±31.5 °C |