| 常用名 | Samuraciclib | CAS号 | 1805833-75-3 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: Samuraciclib (CT7001) is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC50 of 41 nM. Samuraciclib displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC50 of 578 nM), CDK5 and CDK9, respectively. Samuraciclib inhibits the growth of breast cancer cell lines with GI50 values between 0.2-0.3 µM. Samuraciclib has anti-tumor effects[1][2]. 物理化学性质: CAS号:1805833-75-3 常用中文名:Samuraciclib 常用英文名:Samuraciclib 分子式:C22H30N6O 分子量:394.51 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:2-8°C,干燥,密封,避光 |