| 常用名 | CDK12-IN-5 | CAS号 | 2651200-35-8 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: CDK12-IN-5, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC50 of 23.9 nM at high ATP (2 mM). CDK12-IN-5 has no effect on CDK2/Cyclin E (IC50=173 μM) and CDK9/Cyclin T1 (IC50=127 μM) at high ATP (2 mM) (WO2021116178A1)[1]. 物理化学性质: CAS号:2651200-35-8 常用中文名:CDK12-IN-5 常用英文名:CDK12-IN-5 分子式:C18H15F5N8O 分子量:454.36 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |