| 常用名 | MLS1547 | CAS号 | 315698-36-3 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: MLS1547 is a highly efficacious G protein-biased dopamine D2 receptor (D2R) agonist (Ki=1.2 μM). MLS1547 stimulates D2R G protein-mediated signaling (EC50=0.37 μM in a calcium mobilization assay). MLS1547 acts as an antagonist for dopamine (DA)-stimulated β-arrestin recruitment to the D2R (IC50=9.9 μM)[1][2]. 物理化学性质: CAS号:315698-36-3 常用中文名:MLS1547 常用英文名:MLS 1547 分子式:C19H19ClN4O 分子量:354.833 密度:1.4±0.1 g/cm3 沸点:555.8±50.0 °C at 760 mmHg 熔点:N/A 闪点:289.9±30.1 °C 储存条件:-20°C |