| 常用名 | PKUMDL WQ 2201 | CAS号 | 592474-91-4 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: PKUMDL-WQ-2201 is a PHGDH non-NAD+-competing allosteric inhibitor (IC50=35.7 μM). PKUMDL-WQ-2201 also inhibits PHGDH mutants with IC50s of 69 μM (T59A) and >300 μM (T56AK57A), respectively. PKUMDL-WQ-2201 inhibits de novo serine synthesis in cancer cells, and reduces tumor growth[1][2]. 物理化学性质: CAS号:592474-91-4 常用中文名:PKUMDL WQ 2201 常用英文名:PKUMDL WQ 2201 分子式:C15H14ClN3O3S 分子量:351.808 密度:1.4±0.1 g/cm3 沸点:523.5±60.0 °C at 760 mmHg 熔点:N/A 闪点:270.4±32.9 °C |