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4-(2-(2-(二甲基氨基)-2-氧代乙氧基)-2-氧代乙基)苯基4-胍基苯甲酸酯甲磺酸盐

更新时间:2025-08-20 10:35:48 采购访问:51次

常用名 甲磺酸卡莫司他 CAS号 59721-29-8
价格 纯度 98.0%
备货期 10天 库存 现货
 产品详情(用途,包装等)
用途:
Camostat Mesylate(FOY305; FOY-S980) is a trypsin-like protease inhibitorTarget: Trypsin-like proteaseCamostat mesilate (500 mM) inhibits generation of TGF-beta by suppressing plasmin activity and reduces the activity of TGF-beta, which blocks in vitro activation of HSCs [1]. Camostat mesilate (20 mM) combined with insulin results a significant hypoglycemic effect following large intestinal administration. Camostat mesilate (20 mM) is effective in reducing insulin degradation in both small and large intestinal homogenates of rats [2]. Camostat mesilate (2 mM) inhibits MCP-1 and TNF- production in activated rat monocytes. Camostat mesilate (2 mM) inhibits proliferation and MCP-1 production of cultured rat PSCs. Camostat mesilate (1 mg/g) prevents pancreatic atrophy and improves pancreatic exocrine function of rat chronic pancreatitis induced by DBTC. Camostat mesilate (1 mg/g) inhibits chronic inflammation and pancreatic fibrosis induced by DBTC. Camostat mesilate (1 mg/g) inhibits the development of pancreatic fibrosis and PSCs activation in the pancreas induced by DBTC. Camostat mesilate (1 mg/g) suppresses monocytes infiltration and inhibits MCP-1 expression both in serum and in pancreatic tissue [3].
物理化学性质:
CAS号:59721-29-8
常用中文名:甲磺酸卡莫司他
常用英文名:Camostat Mesylate
分子式:C21H26N4O8S
分子量:494.518
密度:N/A
沸点:634.6ºC at 760 mmHg
熔点:150-1550C
闪点:N/A
储存条件:Desiccate at RT

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参考价格:$55/10mM*1mLinDMSO
其他供应商价格:
2025-09-17 4-(2-(2-(二甲基氨基)-2-氧代乙氧基)-2-氧代乙基)苯基4-胍基苯甲酸酯甲磺酸盐
价格:¥需询单
2022-02-19 卡莫他特甲磺酸盐
价格:¥260.9
2017-04-24 甲磺酸卡莫司他
价格:¥需询单
2022-05-12 CaMostat Mesylate
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2021-02-06 Camostat Mesilate
价格:¥889.0
2023-06-26 甲磺酸卡莫司他
价格:¥需询单
2018-03-02 甲磺酸卡莫司他
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2024-05-16 甲磺酸卡莫司他
价格:¥需询单
2024-01-09 Camostat mesilate
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