| 常用名 | HDAC1,2-IN-2 | CAS号 | 937727-03-2 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: A potent, selective HDAC1 and HDAC2 inhibitor with IC50 of 6 nM and 45 nM, respectively; displays highly selectivity over HDAC3 (IC50=7.0 μM), HDAC8 and 11 (IC50=20-25 uM) and no activity on HDACs 4-7; increases lysine 5 of histone H2B (H2BK5) in HCT116 colon carcinoma cells with IC50 of 400 nM, inhibited the cell growth with GI50 of 97 nM; exhibits tumor growth inhibition in HCT116 xenograft mice. 物理化学性质: CAS号:937727-03-2 常用中文名:HDAC1,2-IN-2 常用英文名:HDAC1,2-IN-2 分子式:C23H23N5O3S 分子量:449.529 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |