| 常用名 | PF-6870961 | CAS号 | 2857112-06-0 |
|---|---|---|---|
| 价格 | ¥需询单/100mg ¥需询单/250mg ¥需询单/1g | 纯度 | 98.0% |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: PF-6870961 is an inverse agonist of GHSR1a with Ki values of 73.6 nM (human GHSR), 239 nM (rat GHSR), and 217 nM (dog GHSR), respectively. PF-6870961 inhibits the constitutive GHSR1a-induced IP accumulation with an IC50 value of 300 nM. PF-6870961 also inhibits constitutive GHSR1a β-arrestin mobilization with an IC50 value of 1.10 nM[1]. 物理化学性质: CAS号:2857112-06-0 常用中文名:PF-6870961 常用英文名:PF-6870961 分子式:C29H32N6O2S 分子量:528.67 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |