365996-05-0

• 常用中文名：2-氨基-6,7-二氢噻唑并[5,4-c]吡啶-5(4H)-甲酸叔丁酯
• 常用英文名：tert-butyl 2-amino-6,7-dihydrothiazolo[5,4-c]pyridine-5(4H)-carboxylate
• CAS号：365996-05-0
• 分子式：C₁₁H₁₇N₃O₂S
• 分子量：255.337
• 发布时间：2018-09-05 16:30:00
• 更新时间：2026-07-04 17:04:38
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名称

• 中文名: 2-氨基-6,7-二氢噻唑并[5,4-c]吡啶-5(4H)-甲酸叔丁酯
• 英文名: tert-Butyl 2-amino-6,7-dihydrothiazolo[5,4-c]pyridine-5(4H)-carboxylate
• 中文别名: 2-氨基-6,7-二氢噻唑并[5,4-C]吡啶-5(4H)-甲酸叔丁酯; 5-Boc-2-氨基-4,5,6,7-四氢噻唑并[5,4-c]吡啶; 5-BOC-2-氨基-4,5,6,7-四氢噻唑并[5,4-C]吡啶; 2-氨基-6,7-二氢-4H-噻唑[4,5-C]并吡啶-5-甲酸叔丁酯; 2-氨基-6,7-二氢-4H-噻唑[4,5-c]并吡啶-5-甲酸叔丁酯; 2-氨基-6,7-二氢[1,3]噻唑并[5,4-C]吡啶-5(4H)甲酸叔丁酯; 2-氨基-6,7-二氢噻唑并[5,4-C]嘧啶-5(4H)羧酸叔丁酯; 2-氨基-6,7-二氢[1,3]三唑[5,4-C]吡啶-5(4H)-羧酸叔丁酯
• 英文别名: tert-butyl 2-amino-6; tert-butyl 2-amino-6,7-dihydro[1,3]thiazolo[5,4-c]pyridine-5(4H)-carboxylate; 2-Amino-5-Boc-6,7-dihydro-4H-thiazolo-[5,4,c]pyridine; tert-butyl 2-amino-6.7-dihydrothiazolo[5.4-c]pyridine-5(4H)-cb; tert-butyl 2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridine-5-cboxylate; tert-butyl 2-amino-6,7-dihydro-4H-thiazolo[5,4-c]pyridine-5-cboxylate; tert-Butyl 2-amino-6,7-dihydro[1,3]thiazolo[5,4-c]pyridine-5(4H)-cboxylate, 2-Amino-5-(tert-butoxycbonyl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridine; Thiazolo[5,4-c]pyridine-5(4H)-carboxylic acid, 2-amino-6,7-dihydro-, 1,1-dimethylethyl ester; tert-butyl 2-amino-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carboxylate; tert-butyl 2-amino-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-cboxylate; Thiazolo[5,4-c]pyridine-5(4H)-cboxylic acid, 2-amino-6,7-dihydro-, 1,1-dimethylethyl ester; 2-Amino-6,7-dihydro-4H-thiazolo[5,4-c]pyridine-5-cboxylic acid tert-butyl ester; 2-Amino-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridine, N5-BOC protected; 2-Methyl-2-propanyl 2-amino-6,7-dihydro[1,3]thiazolo[5,4-c]pyridine-5(4H)-carboxylate; 4-c]pyridine-5(4H)-cboxylate; 7-dihydrothiazolo[5; ENCHEM TERT-BUTYL 2-AMINO-6,7-DIHYDRO[1,3]THIAZOLO[5,4-C]PYRIDINE-5(4H)-CBOXYLATE 365-0; tert-butyl 2-amino-6,7-dihydro[1,3]thiazolo[5,4-c]pyridine-5; 4,5,6,7-tetrahydro-5-Boc-thiazolo[5,4-c]pyridin-2-amine; 1,1-Dimethylethyl 2-amino-6,7-dihydrothiazolo[5,4-c]pyridine-5(4H)-cboxylate; 5-Boc-2-Amino-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine

物化性质

• 密度: 1.3±0.1 g/cm3
• 沸点: 412.8±45.0 °C at 760 mmHg
• 分子式: C₁₁H₁₇N₃O₂S
• 分子量: 255.337
• 闪点: 203.4±28.7 °C
• 精确质量: 255.104141
• PSA: 96.69000
• LogP: 1.11
• 蒸汽压: 0.0±1.0 mmHg at 25°C
• 折射率: 1.592
• 储存条件: 2-8°C

安全

• 危害码 (欧洲): Xi
• 海关编码: 2934999090

合成路线

420-04-2 207691-65-4 ~% 365996-05-0

文献：EP1405852 A1, ; Page 65 ; EP 1405852 A1

60-35-5 79099-07-3 ~% 365996-05-0

文献：WO2008/86047 A1, ; Page/Page column 127-128 ; WO 2008/086047 A1

420-04-2 79099-07-3 ~62% 365996-05-0

文献：Haginoya, Noriyasu; Komoriya, Satoshi; Osanai, Ken; Yoshino, Toshiharu; Nagata, Tsutomu; Nagamochi, Masatoshi; Muto, Ryo; Yamaguchi, Mitsuhiro; Nagahara, Takayasu; Kanno, Hideyuki Heterocycles, 2004 , vol. 63, # 7 p. 1555 - 1561

420-04-2 ~% 365996-05-0

文献：EP1577301 A1, ; Page/Page column 72 ;

17356-08-0 188869-05-8 ~% 365996-05-0

文献：WO2006/108709 A1, ; Page/Page column 69 ; WO 2006/108709 A1

24424-99-5 97817-23-7 ~% 365996-05-0

文献：GRAUERT, Matthias; BISCHOFF, Daniel; DAHMANN, Georg; KUELZER, Raimund; RUDOLF, Klaus; WELLENZOHN, Bernd Patent: US2013/150341 A1, 2013 ; Location in patent: Paragraph 0179; 0180; 0181 ;

24424-99-5 17356-08-0 188869-05-8 ~% 365996-05-0

文献：WO2007/95124 A2, ; Page/Page column 63-64 ;

79099-07-3 ~% 365996-05-0

文献：WO2004/43968 A1, ; Page 22 ; WO 2004/043968 A1

41661-47-6 ~% 365996-05-0

文献：WO2013/83741 A1, ;

上下游产品

上游产品  8
420-04-2 207691-65-4 60-35-5 79099-07-3
188869-05-8 24424-99-5 97817-23-7 41661-47-6
下游产品  3
365996-06-1 365996-07-2 143150-92-9

海关

海关编码	2934999090
中文概述	2934999090. 其他杂环化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%
申报要素	品名, 成分含量, 用途
Summary	2934999090. other heterocyclic compounds. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%