Cholesterol 24-hydroxylase-IN-2

• 常用名: Cholesterol 24-hydroxylase-IN-2
• 英文名: Cholesterol 24-hydroxylase-IN-2
• CAS号: 1613481-52-9
• 分子量: 354.42
• 密度: N/A
• 沸点: N/A
• 分子式: C₂₀H₂₃FN₄O
• 熔点: N/A
• 闪点: N/A

Cholesterol 24-hydroxylase-IN-2用途

Cholesterol 24-Hydroxylase-IN-2 是胆固醇 24-羟化酶(CH24H 或 CYP46A1)的抑制剂,IC50 为 5.4 nM。 胆固醇 24-羟化酶-IN-2 可用于哺乳动物胆固醇 24-羟化酶的成像。

Cholesterol 24-hydroxylase-IN-2名称

• 英文名: Cholesterol 24-hydroxylase-IN-2

Cholesterol 24-hydroxylase-IN-2生物活性

• 描述: Cholesterol 24-Hydroxylase-IN-2 是胆固醇 24-羟化酶(CH24H 或 CYP46A1)的抑制剂,IC50 为 5.4 nM。 胆固醇 24-羟化酶-IN-2 可用于哺乳动物胆固醇 24-羟化酶的成像。
• 相关类别:
  信号通路 >> 代谢酶/蛋白酶 >> 细胞色素P450
  研究领域 >> 其他
• 参考文献:

  [1]. Koike Tatsuki, et al. Preparation of arylpiperidines and arylpiperazines as radiolabeled compounds for use in imaging of cholesterol 24-hydroxylase. World Intellectual Property Organization, WO2015190613 A1 2015-12-17

Cholesterol 24-hydroxylase-IN-2物理化学性质

• 分子式: C₂₀H₂₃FN₄O
• 分子量: 354.42

Cholesterol 24-hydroxylase-IN-2靶点实验

查看更多实验

实验名称：Inhibitory Assay from US Patent US9963443: "Radiolabeled compounds" 来源：BindingDB 靶标：N/A External Id：BindingDB_3165_1

实验名称：Inhibition of human CH24H expressed in Freestyle-293 cells assessed as reduction in 2... 来源：ChEMBL 靶标：Cholesterol 24-hydroxylase External Id：CHEMBL4477128

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