(S)-Cipepofol

更新时间：2025-08-27 10:11:39

(S)-Cipepofol用途

(S)-Cipepofol 是 Cipepofol (HY-116152 ) 的非活性异构体。Cipepofol (HSK3486) 是一种促进睡眠活性分子,是一种γ-氨基丁酸 (GABA) 受体增强剂。

英文名	(S)-Cipepofol

描述	(S)-Cipepofol 是 Cipepofol (HY-116152 ) 的非活性异构体。Cipepofol (HSK3486) 是一种促进睡眠活性分子,是一种γ-氨基丁酸 (GABA) 受体增强剂。
相关类别	信号通路 >> 跨膜转运 >> GABA受体研究领域 >> 神经疾病信号通路 >> 神经信号通路 >> GABA受体
参考文献	[1]. Li X, et al. Safety, Pharmacokinetics, and Pharmacodynamics of a Single Bolus of the γ-aminobutyric Acid (GABA) Receptor Potentiator HSK3486 in Healthy Chinese Elderly and Non-elderly. Front Pharmacol. 2021;12:735700. Published 2021 Aug 27.

分子式	C₁₄H₂₀O
分子量	204.31

实验名称：Displacement of [35S]TBPS from GABAA receptor in Wistar rat cerebral cortex membranes...
来源：ChEMBL
靶标：N/A
External Id：CHEMBL4043673

实验名称：Displacement of [35S]TBPS from GABAA receptor in Wistar rat cerebral cortex membranes...
来源：ChEMBL
靶标：N/A
External Id：CHEMBL4043674

实验名称：Displacement of [35S]TBPS from GABAA receptor in Wistar rat cerebral cortex membranes...
来源：ChEMBL
靶标：N/A
External Id：CHEMBL4043672

实验名称：Toxicity in iv dosed ICR mouse administered 7 to 8 doses at 10 secs for each dose
来源：ChEMBL
靶标：Mus musculus
External Id：CHEMBL4043685

实验名称：Anesthetic activity in iv dosed ICR mouse assessed as dose required to produce 10 min...
来源：ChEMBL
靶标：Mus musculus
External Id：CHEMBL4043686

实验名称：Anesthetic activity in iv dosed ICR mouse assessed as recovery time of righting refle...
来源：ChEMBL
靶标：Mus musculus
External Id：CHEMBL4043683

实验名称：Anesthetic activity in iv dosed ICR mouse assessed as loss of righting reflex adminis...
来源：ChEMBL
靶标：Mus musculus
External Id：CHEMBL4043684

实验名称：Anesthetic activity in iv dosed ICR mouse assessed as onset time for loss of righting...
来源：ChEMBL
靶标：Mus musculus
External Id：CHEMBL4043681

实验名称：Anesthetic activity in iv dosed ICR mouse assessed as anesthetic duration time admini...
来源：ChEMBL
靶标：Mus musculus
External Id：CHEMBL4043682

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