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IU1-248

更新时间:2024-01-10 16:33:26

IU1-248结构式
IU1-248结构式
品牌特惠专场
常用名 IU1-248 英文名 IU1-248
CAS号 2307472-03-1 分子量 337.42
密度 N/A 沸点 N/A
分子式 C20H23N3O2 熔点 N/A
MSDS N/A 闪点 N/A

 IU1-248用途


IU1-248是IU1的衍生物,是一种有效的选择性USP14抑制剂,IC50为0.83 μM。

 IU1-248名称

英文名 IU1-248

 IU1-248生物活性

描述 IU1-248是IU1的衍生物,是一种有效的选择性USP14抑制剂,IC50为0.83 μM。
相关类别
体外研究 IU1-248的IC50值为0.83 与IU1-47(IC50=0.68μM)相当,效力是IU1(IC50=12.25μM)的10倍[1]。
参考文献

[1]. Yiwei Wang, et al. Small molecule inhibitors reveal allosteric regulation of USP14 via steric blockade. Cell Res. 2018 Dec;28(12):1186-1194.

 IU1-248物理化学性质

分子式 C20H23N3O2
分子量 337.42
储存条件 2-8°C
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IU1-248价格

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