2-([1,1'-联苯]-4-基)-N-(吡啶-2-基)乙酰胺

• 常用名: 2-([1,1'-联苯]-4-基)-N-(吡啶-2-基)乙酰胺
• 英文名: [1,1'-Biphenyl]-4-acetamide,N-2-pyridinyl
• CAS号: 51484-40-3
• 分子量: 288.34300
• 密度: 1.192g/cm3
• 沸点: 549ºC at 760 mmHg
• 分子式: C₁₉H₁₆N₂O
• 熔点: N/A
• 闪点: 285.8ºC

用途

二苯吡酰胺(Z-876)是一种双苯乙醇衍生物,具有显著的抗炎、镇痛、解热和尿酸特性。二苯吡酰胺具有抗血小板聚集活性[1]。

名称

• 中文名: 联苯吡胺
• 英文名: difenpiramide

生物活性

• 描述: 二苯吡酰胺(Z-876)是一种双苯乙醇衍生物,具有显著的抗炎、镇痛、解热和尿酸特性。二苯吡酰胺具有抗血小板聚集活性[1]。
• 相关类别:
  信号通路 >> 其他 >> 其他
  研究领域 >> 炎症/免疫
• 参考文献:

  [1]. Caliari S, et al. Pharmacological properties of the anti-inflammatory agent pyridyl-biphenylyl-acetamide (diphenpyramide). Arzneimittelforschung. 1977;27(11):2086-2093.

  [2]. Gugliotta L, et al. Farmaci antiinfiammatori e attività antiaggregante piastrinica: la difenpiramide [Anti-inflammatory drugs and platelet anti-aggregation activity: difenpiramide]. G Clin Med. 1976;57(11-12):408-415.

物理化学性质

• 密度: 1.192g/cm3
• 沸点: 549ºC at 760 mmHg
• 分子式: C₁₉H₁₆N₂O
• 分子量: 288.34300
• 闪点: 285.8ºC
• 精确质量: 288.12600
• PSA: 41.99000
• LogP: 4.00280
• 折射率: 1.645
• 储存条件: 室温

毒性和生态

安全信息

• 海关编码: 2933399090

海关

• 海关编码: 2933399090
• 中文概述: 2933399090. 其他结构含非稠合吡啶环的化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%
• 申报要素: 品名, 成分含量, 用途, 乌洛托品请注明外观, 6－己内酰胺请注明外观, 签约日期
• Summary: 2933399090. other compounds containing an unfused pyridine ring (whether or not hydrogenated) in the structure. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

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英文别名

• Z-876
• 2-Biphenylyl-N-pyridylacetamide
• 2-(4-phenylphenyl)-N-pyridin-2-ylacetamide
• Pyridyl-biphenylyl-acetamide
• Difenax
• Acetamide,2-biphenylyl-N-pyridyl
• Difenpiramide
• Diphenpyramide