3-Phenylacetylamino-2,6-piperidinedione

• 常用名: 3-Phenylacetylamino-2,6-piperidinedione
• 英文名: (rac)-Antineoplaston A10
• CAS号: 77658-84-5
• 分子量: 246.26
• 密度: 1.27 g/cm3
• 沸点: 571.2ºC at 760 mmHg
• 分子式: C₁₃H₁₄N₂O₃
• 熔点: N/A
• 闪点: N/A

用途

(rac)-Antineoplaston A10 是(rac)-Antineoplaston A10 的消旋体。Antineoplaston A10是 Ras 的一个抑制剂,可用于治疗胶质瘤、淋巴瘤、星形细胞瘤和乳腺癌。

3-Phenylacetylamino-2,6-piperidinedione名称

• 中文名: 1,1'-二甲基-4,4'-联吡啶翁盐
• 英文名: Antineoplaston A10
• 中文别名: 3-苯基乙酰氨基-2,6-哌啶二酮 | 抗瘤酮 A10

3-Phenylacetylamino-2,6-piperidinedione生物活性

• 描述: (rac)-Antineoplaston A10 是(rac)-Antineoplaston A10 的消旋体。Antineoplaston A10是 Ras 的一个抑制剂,可用于治疗胶质瘤、淋巴瘤、星形细胞瘤和乳腺癌。
• 相关类别:
  研究领域 >> 癌症
  信号通路 >> 其他 >> 其他
• 参考文献:

  [1]. Qu XJ, et al. Induction of apoptosis in human hepatocellular carcinoma cells by synthetic antineoplaston A10. Anticancer Res. 2007 Jul-Aug;27(4B):2427-31.

3-Phenylacetylamino-2,6-piperidinedione物理化学性质

• 密度: 1.27 g/cm3
• 沸点: 571.2ºC at 760 mmHg
• 分子式: C₁₃H₁₄N₂O₃
• 分子量: 246.26
• 精确质量: 246.10000
• PSA: 75.27000
• LogP: 0.87020
• InChIKey: OQGRFQCUGLKSAV-UHFFFAOYSA-N
• SMILES: O=C1CCC(NC(=O)Cc2ccccc2)C(=O)N1
• 外观性状: 固体
• 折射率: 1.584
• 储存条件: 2-8°C，密封，干燥

3-Phenylacetylamino-2,6-piperidinedione安全信息

• 危害码 (欧洲): Xi

3-Phenylacetylamino-2,6-piperidinedione靶点实验

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3-Phenylacetylamino-2,6-piperidinedione英文别名

• 3-Phenylacetylamino-2,6-piperidinedione