Synthetic Communications®

Cu (OAc) 2-catalyzed N-arylation of sulfonamides with arylboronic acids or trimethoxy (phenyl) silane

C Pan, J Cheng, H Wu, J Ding, M Liu

Index: Pan, Changduo; Cheng, Jiang; Wu, Huayue; Ding, Jinchang; Liu, Miaochang Synthetic Communications, 2009 , vol. 39, # 12 p. 2082 - 2092

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Citation Number: 14

Abstract

N-Arylsulfonamides have long been the subjects of pharmaceutical interest because of their potential biological activities. [ 1 1. ( a ) Harter , WG ; Albrect , H. ; Brady , K. ; Caprathe , B. ; Dunbar , J. ; Gilmore , J. ; Hays , S. ; Kostlan , CR ; Lunney , B. ; Walker , N. The design and synthesis of sulfonamides as caspase-1 inhibitors . Bioorg. Med. Chem. Lett. 2004 , 14 , 809 – 812 ; ( b ) Reddy , NSM ; Mallireddigari , R. ; Cosenza , KG ; Bell , SC ; Reddy , EP ; Reddy , MVR ...