The Journal of organic chemistry

Scope and limitations of the Pd/BINAP-catalyzed amination of aryl bromides

JP Wolfe, SL Buchwald

Index: Itier,J.; Casadevall,A. Bulletin de la Societe Chimique de France, 1969 , p. 2342 - 2355

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Citation Number: 477

Abstract

... weak bases such as alkali metal carbonates and phosphates, 2e,j as well as organic bases such as tertiary amines and DBU. These generally gave poorer results in the amination reactions. The activated substrate 4-bromobenzonitrile was efficiently coupled with p-toluidine in ...