Palladium??Catalyzed Direct Arylations of Heteroarenes with Tosylates and Mesylates

L Ackermann, A Althammer…

Index: Ackermann, Lutz; Althammer, Andreas; Fenner, Sabine Angewandte Chemie - International Edition, 2009 , vol. 48, # 1 p. 201 - 204

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Citation Number: 235

Abstract

Palladium-catalyzed cross-coupling reactions between organic halides or triflates and organometallic reagents are among the most important tools for regioselective C (sp2) À C (sp2) bond formations.[1–3] Particularly, their applications to heteroaromatic substrates sets the stage for novel routes to substituted heterocycles, which are valuable substructures of compounds having activities that are relevant to material or biological sciences.[4] The ...

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