Synlett

Copper promoted aryl/saturated heterocyclic CN bond cross-coupling with arylboronic acid and arylstannane

PYS Lam, CG Clark, S Saubern, J Adams, KM Averill…

Index: Lam, Patrick Y.S.; Clark, Charles G.; Saubern, Simon; Adams, Jessica; Averill, Kristin M.; Chan, Dominic M. T.; Combs, Andrew Synlett, 2000 , # 5 p. 674 - 676

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Citation Number: 135

Abstract

Abstract: Arylboronic acid/cupric acetate arylation of NH containing saturated heterocycles has been explored and found to give good yields of the cross-coupled products. Phenyltrimethylstannane is also found to arylate NH containing heterocycles. Key words: N- arylation, copper (II) acetate, stannane, boronic acid, cross-coupling